6uil A 2.85 BS01 FKS A 1 D94 P134 H136 H137 F146 D174 H176 W205 E274 E304 G305 Y307 D93 P133 H135 H136 F145 D173 H175 W204 E273 E303 G304 Y306 3.5.1.48,3.5.1.62 0005634,0005737,0008270,0016236,0016787,0019213,0033558,0035825,0036269,0040029,0046872,0047609,0047611,0090043,0106047,0106048 -logKd/Ki=7.10, IC50=80nM F1QCV2 31746596 701 ASGSALIFDEEMSRYKLLWTDPACEIEVPERLTVSYEALRTHGLAQRCKAVPVRQATEQEILLAHSEEYLEAVKQTPGMNVEELMAFSKKYNDVYFHQNIYHCAKLAAGATLQLVDSVMKREVRNGMALVRPPGHHSQRSAANGFCVFNNVAFAALYAKKNYNLNRILIVDWDVHHGQGIQYCFEEDPSVLYFSWHRYEHQSFWPNLPESDYSSVGKGKGSGFNINLPWNKVGMTNSDYLAAFFHVLLPVAYEFDPELVIVSAGFDSAIGDPEGEMCALPEIFAHLTHLLMPLAAGKMCVVLEGGYNLTSLGQSVCQTVHSLLGDPTPRISGLGTACDSALESIQNVRNVQSSYWSSFKHLAQSVRTVVVPPPGVELTLPKNCQHSISESTAKEVQRIRDKHFDQNILRSLGNIISVLDRMMVCNGCVVVSDLSVSVQCALQHALTEPAERVLVVYVGDGELPVKTNDGKVFLVQICTKETEDKCVNRLTLCGESLTAGFMQALLGLILPVAYEFNPALVLGIVEETRLMRVWGHMTCLIQGLARGRMLTLLQDKDLLELTVSALSGASISPLGPAPKPEDVEMMEKQRQRLQERWGLLRCTVSESW 6uil A 2.85 BS02 ZN A 1 D174 H176 D267 D173 H175 D266 3.5.1.48,3.5.1.62 0005634,0005737,0008270,0016236,0016787,0019213,0033558,0035825,0036269,0040029,0046872,0047609,0047611,0090043,0106047,0106048 F1QCV2 31746596 704 ASGSALIFDEEMSRYKLLWTDPACEIEVPERLTVSYEALRTHGLAQRCKAVPVRQATEQEILLAHSEEYLEAVKQTPGMNVEELMAFSKKYNDVYFHQNIYHCAKLAAGATLQLVDSVMKREVRNGMALVRPPGHHSQRSAANGFCVFNNVAFAALYAKKNYNLNRILIVDWDVHHGQGIQYCFEEDPSVLYFSWHRYEHQSFWPNLPESDYSSVGKGKGSGFNINLPWNKVGMTNSDYLAAFFHVLLPVAYEFDPELVIVSAGFDSAIGDPEGEMCALPEIFAHLTHLLMPLAAGKMCVVLEGGYNLTSLGQSVCQTVHSLLGDPTPRISGLGTACDSALESIQNVRNVQSSYWSSFKHLAQSVRTVVVPPPGVELTLPKNCQHSISESTAKEVQRIRDKHFDQNILRSLGNIISVLDRMMVCNGCVVVSDLSVSVQCALQHALTEPAERVLVVYVGDGELPVKTNDGKVFLVQICTKETEDKCVNRLTLCGESLTAGFMQALLGLILPVAYEFNPALVLGIVEETRLMRVWGHMTCLIQGLARGRMLTLLQDKDLLELTVSALSGASISPLGPAPKPEDVEMMEKQRQRLQERWGLLRCTVSESW