6s9b A 3.25 BS01 L1H A 1 L718 A743 K745 E762 M790 Q791 M793 P794 G796 L844 T854 L22 A47 K49 E63 M91 Q92 M94 P95 G97 L145 T155 D837 R841 N842 D855 D138 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=5.68, IC50=2100nM P00533 31689114 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKEATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPDDVVDADEYLIP