6qxs A 2.88 BS01 UFP B 1 R177 R178 R156 R157 E59 W81 Y145 C197 R217 D220 E59 W81 Y124 C176 R196 D199 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 -logKd/Ki=7.13, Ki=74nM Q834R3 30935102 401 MEEAYLALGKKILEEGHFKEDRTGTGTYSLFGYQMRFDLAKGFPLLTTKRVPFGLIKSELLWFLKGDTNIRYLLERNNHIWDEWAFERYVKSADYQGEEHQKFCDAILNDAEFAEKYGELGNIYGAQWRHWETKDGSFIDQLANVIEMIKTNPDSRRLIVSAWNPEDVPSMALPPCHTMFQFYVNEGKLSCQLYQRSADVFLGVPFNIASYALLTHLIAHETGLEVGEFVHTLGDAHLYQNHVEQMQEQLSREVRSFPTLVLNPDKASVFDFDMEDIKVEGYDPHPTIKAPI 6qxs B 2.88 BS01 UFP B 1 R22 Y145 C197 H198 R217 S218 D220 N228 H258 Y260 R22 Y145 C197 H198 R217 S218 D220 N228 H258 Y260 E59 W81 Y145 C197 R217 D220 E59 W81 Y145 C197 R217 D220 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 -logKd/Ki=7.13, Ki=74nM Q834R3 30935102 401 MEEAYLALGKKILEEGHFKEDRTGTGTYSLFGYQMRFDLAKGFPLLTTKRVPFGLIKSELLWFLKGDTNIRYLLERNNHIWDEWAFERYVKSADYQGPDMTDFGHRVLQDPAFAEQYKEEHQKFCDAILNDAEFAEKYGELGNIYGAQWRHWETKDGSFIDQLANVIEMIKTNPDSRRLIVSAWNPEDVPSMALPPCHTMFQFYVNEGKLSCQLYQRSADVFLGVPFNIASYALLTHLIAHETGLEVGEFVHTLGDAHLYQNHVEQMQEQLSREVRSFPTLVLNPDKASVFDFDMEDIKVEGYDPHPTIKAPIAV 6qxs B 2.88 BS02 FFO B 1 I80 W81 W84 D220 L223 F227 I313 I80 W81 W84 D220 L223 F227 I313 E59 W81 Y145 C197 R217 D220 E59 W81 Y145 C197 R217 D220 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Q834R3 30935102 403 MEEAYLALGKKILEEGHFKEDRTGTGTYSLFGYQMRFDLAKGFPLLTTKRVPFGLIKSELLWFLKGDTNIRYLLERNNHIWDEWAFERYVKSADYQGPDMTDFGHRVLQDPAFAEQYKEEHQKFCDAILNDAEFAEKYGELGNIYGAQWRHWETKDGSFIDQLANVIEMIKTNPDSRRLIVSAWNPEDVPSMALPPCHTMFQFYVNEGKLSCQLYQRSADVFLGVPFNIASYALLTHLIAHETGLEVGEFVHTLGDAHLYQNHVEQMQEQLSREVRSFPTLVLNPDKASVFDFDMEDIKVEGYDPHPTIKAPIAV 6qxs C 2.88 BS01 UFP D 1 R177 R178 R156 R157 E59 W81 Y145 C197 R217 D220 E59 W81 Y124 C176 R196 D199 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Q834R3 30935102 401 MEEAYLALGKKILEEGHFKEDRTGTGTYSLFGYQMRFDLAKGFPLLTTKRVPFGLIKSELLWFLKGDTNIRYLLERNNHIWDEWAFERYVKSADYQGEEHQKFCDAILNDAEFAEKYGELGNIYGAQWRHWETKDGSFIDQLANVIEMIKTNPDSRRLIVSAWNPEDVPSMALPPCHTMFQFYVNEGKLSCQLYQRSADVFLGVPFNIASYALLTHLIAHETGLEVGEFVHTLGDAHLYQNHVEQMQEQLSREVRSFPTLVLNPDKASVFDFDMEDIKVEGYDPHPTIKAPI 6qxs D 2.88 BS01 UFP D 1 R22 Y145 C197 H198 R217 S218 D220 H258 Y260 R22 Y145 C197 H198 R217 S218 D220 H258 Y260 E59 W81 Y145 C197 R217 D220 E59 W81 Y145 C197 R217 D220 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Q834R3 30935102 401 MEEAYLALGKKILEEGHFKEDRTGTGTYSLFGYQMRFDLAKGFPLLTTKRVPFGLIKSELLWFLKGDTNIRYLLERNNHIWDEWAFERYVKSADYQGPDMTDFGHRVLQDPAFAEQYKEEHQKFCDAILNDAEFAEKYGELGNIYGAQWRHWETKDGSFIDQLANVIEMIKTNPDSRRLIVSAWNPEDVPSMALPPCHTMFQFYVNEGKLSCQLYQRSADVFLGVPFNIASYALLTHLIAHETGLEVGEFVHTLGDAHLYQNHVEQMQEQLSREVRSFPTLVLNPDKASVFDFDMEDIKVEGYDPHPTIKAPIAV 6qxs D 2.88 BS02 FFO D 1 I80 W81 W84 D220 I313 A314 I80 W81 W84 D220 I313 A314 E59 W81 Y145 C197 R217 D220 E59 W81 Y145 C197 R217 D220 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Q834R3 30935102 403 MEEAYLALGKKILEEGHFKEDRTGTGTYSLFGYQMRFDLAKGFPLLTTKRVPFGLIKSELLWFLKGDTNIRYLLERNNHIWDEWAFERYVKSADYQGPDMTDFGHRVLQDPAFAEQYKEEHQKFCDAILNDAEFAEKYGELGNIYGAQWRHWETKDGSFIDQLANVIEMIKTNPDSRRLIVSAWNPEDVPSMALPPCHTMFQFYVNEGKLSCQLYQRSADVFLGVPFNIASYALLTHLIAHETGLEVGEFVHTLGDAHLYQNHVEQMQEQLSREVRSFPTLVLNPDKASVFDFDMEDIKVEGYDPHPTIKAPIAV