6pt0 R 3.2 BS01 WI5 R 1 F87 S90 F94 I110 T114 F183 P184 Y190 L191 W194 F66 S69 F73 I89 T93 F162 P163 Y169 L170 W173 ? 0001975,0004930,0004949,0005515,0005737,0005783,0005886,0006954,0006955,0007186,0007187,0007189,0016020,0019222,0030425,0030595,0031234,0032229,0032496,0033004,0038171,0042995,0043025,0043204,0045211,0045759,0099553 Ki=2.1nM, EC50=24.6nM, IC50=3.4nM P34972 32004460 401 MKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKK 6pt0 R 3.2 BS02 CLR R 1 Q276 F283 Q255 F262 ? 0001975,0004930,0004949,0005515,0005737,0005783,0005886,0006954,0006955,0007186,0007187,0007189,0016020,0019222,0030425,0030595,0031234,0032229,0032496,0033004,0038171,0042995,0043025,0043204,0045211,0045759,0099553 P34972 32004460 403 MKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKK 6pt0 R 3.2 BS03 CLR R 2 I129 L133 L144 I108 L112 L123 ? 0001975,0004930,0004949,0005515,0005737,0005783,0005886,0006954,0006955,0007186,0007187,0007189,0016020,0019222,0030425,0030595,0031234,0032229,0032496,0033004,0038171,0042995,0043025,0043204,0045211,0045759,0099553 P34972 32004460 404 MKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKK 6pt0 R 3.2 BS04 CLR R 3 G210 L213 W214 G189 L192 W193 ? 0001975,0004930,0004949,0005515,0005737,0005783,0005886,0006954,0006955,0007186,0007187,0007189,0016020,0019222,0030425,0030595,0031234,0032229,0032496,0033004,0038171,0042995,0043025,0043204,0045211,0045759,0099553 P34972 32004460 406 MKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKK