6n78 A 1.83 BS01 KEP A 1 L881 G882 E883 G887 V889 A906 M956 L959 E966 R1007 L1010 G1020 D1021 L16 G17 E18 G22 V24 A41 M81 L84 E91 R132 L135 G145 D146 D1003 A1005 R1007 N1008 D1021 D128 A130 R132 N133 D146 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.21nM -logKd/Ki=9.68, Ki=0.21nM P23458 30981576 1201 DPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK