6mzw A 2.2 BS01 TZ0 A 1 L484 G485 C488 V492 A512 K514 E531 M535 I545 Y563 A564 L630 D641 F642 L21 G22 C25 V29 A49 K51 E68 M72 I82 Y100 A101 L165 D176 F177 D623 R627 N628 D641 D158 R162 N163 D176 2.7.10.1 0004672,0004713,0005007,0005524,0006468 -logKd/Ki=8.41, IC50=3.9nM IC50=3.6nM P11362 30600916 801 ELPEDPRWELPRDRLVLGKPLGEGCFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPGLEYSYNPSPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 6mzw B 2.2 BS01 TZ0 B 1 L484 G485 A512 K514 M535 A564 L630 D641 F642 L22 G23 A43 K45 M66 A95 L146 D157 F158 D623 R627 N628 D641 D139 R143 N144 D157 2.7.10.1 0004672,0004713,0005007,0005524,0006468 IC50=3.6nM P11362 30600916 801 YELPEDPRWELPRDRLVLGKPLGQVVLAEAIGLDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTS