6mo5 A 1.851 BS01 JWP A 1 L18 H19 M62 E77 H78 T190 F191 G192 F193 I197 G209 S210 H237 D241 H264 L23 H24 M67 E82 H83 T194 F195 G196 F197 I201 G213 S214 H241 D245 H268 3.5.1.108 0006796,0008759,0009245,0016787,0019637,0046872,0103117,1901135 ic50=0.3nM -logKd/Ki=9.52, IC50=0.3nM P47205 31283109 301 HHHHATIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFCRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFVRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP 6mo5 A 1.851 BS02 MG A 1 H78 H237 D241 H83 H241 D245 3.5.1.108 0006796,0008759,0009245,0016787,0019637,0046872,0103117,1901135 P47205 31283109 302 HHHHATIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFCRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFVRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP