6m4u A 2.2 BS01 RAP A 1 Y27 F37 D38 F47 Q54 E55 V56 I57 W60 Y83 I92 Y27 F37 D38 F47 Q54 E55 V56 I57 W60 Y83 I92 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,1902991,1990000,1990425 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 32747768 201 MGVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 6m4u B 2.2 BS01 RAP A 1 L2031 E2032 S2035 F2039 Y2105 F2108 L11 E12 S15 F19 Y85 F88 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 32747768 201 ILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRISK 6m4u B 2.2 BS02 ZN B 1 H2028 E2032 H8 E12 2.7.11.1 0044877 P42345 32747768 2201 ILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRISK 6m4u B 2.2 BS03 ZN B 2 D2077 H2106 D57 H86 2.7.11.1 0044877 P42345 32747768 2202 ILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRISK 6m4u E 2.2 BS01 RAP E 1 Y27 F37 D38 F47 E55 V56 I57 W60 Y83 I92 Y29 F39 D40 F49 E57 V58 I59 W62 Y85 I94 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,1902991,1990000,1990425 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 32747768 201 GSMGVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 6m4u F 2.2 BS01 RAP E 1 L2031 E2032 S2035 F2039 L2098 D2102 Y2105 F2108 L13 E14 S17 F21 L80 D84 Y87 F90 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 32747768 201 GSILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRISK 6m4u F 2.2 BS02 ZN F 1 H2028 E2032 H10 E14 2.7.11.1 0044877 P42345 32747768 2201 GSILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRISK 6m4u F 2.2 BS03 ZN F 2 D2077 H2106 D59 H88 2.7.11.1 0044877 P42345 32747768 2205 GSILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRISK