6k1q A 2.7 BS01 D2U A 1 D147 H150 N158 K161 P178 Q181 K182 S184 V185 F240 Y281 W336 L339 R343 A375 S376 S379 D57 H60 N68 K71 P88 Q91 K92 S94 V95 F144 Y185 W343 L346 R350 A382 S383 S386 3.2.1.17 0003796,0004930,0007186,0016020,0016998 -logKd/Ki=7.46, IC50=35nM P00720,P24530 31263780 1201 QGPIEIKETFKYINTVVSCLVFVLGIIGNSTLLYIIYKNKCMRNGPNILIASLALGDLLHIVIDIPINVYKLLAEDWPFGAEMCKLVPFIQKASVGITVLSLCALSIDRYRAVASWSVPKWTAVEIVLIWVVSVVLAVPEAIGFDIITMDYKGSYLRICLLHPVQKTAFMQFYATAKDWWLFSFYFCLPLAITAFFYTLMTCEMLRKNIFEMLRIDEGAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYLNDHLKQRREVAKTVFCLVLVFALCWLPLHLARILKLTLYNQNDPNRCELLSFLLVLDYIGINMASLNSCANPIALYLVSKRFKNAFKSALCC