6hsk A 2.096 BS01 ZN A 1 D178 H180 D267 D165 H167 D254 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031397,0031647,0032204,0033558,0040029,0046872,0051879,0140297,0160008,0160009 Q9BY41 30347148 401 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTISGDRLGCFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 6hsk A 2.096 BS02 GOK A 1 H142 H143 G151 F152 D178 H180 G206 F208 P209 Y306 H129 H130 G138 F139 D165 H167 G193 F195 P196 Y293 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031397,0031647,0032204,0033558,0040029,0046872,0051879,0140297,0160008,0160009 -logKd/Ki=7.03, IC50=93nM IC50=64nM, Ki=24nM, Kd=23nM Q9BY41 30347148 404 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTISGDRLGCFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 6hsk B 2.096 BS01 ZN B 1 D178 H180 D267 D165 H167 D254 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031397,0031647,0032204,0033558,0040029,0046872,0051879,0140297,0160008,0160009 Q9BY41 30347148 401 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTISGDRLGCFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 6hsk B 2.096 BS02 GOK B 1 H142 H143 G151 F152 D178 H180 G206 F208 P209 Y306 H129 H130 G138 F139 D165 H167 G193 F195 P196 Y293 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031397,0031647,0032204,0033558,0040029,0046872,0051879,0140297,0160008,0160009 IC50=64nM, Ki=24nM, Kd=23nM Q9BY41 30347148 404 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTISGDRLGCFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV