6hhh A 2.7 BS01 G4Q A 1 E17 W80 T82 I84 E85 L210 T211 L264 K268 Y272 D292 C296 K297 E16 W76 T78 I80 E81 L161 T162 L215 K219 Y223 D243 C247 K248 D274 K276 N279 D292 T312 D225 K227 N230 D243 T252 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035556,0035655,0035924,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043154,0043161,0043276,0043325,0043488,0043491,0043536,0044024,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060709,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1904263,1905552,1990090,1990418,2000010,2000074,2000402,2001240,2001243 -logKd/Ki=7.17, Ki=67.1nM P31749 30996949 501 SDVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDVEAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGLKKRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFD