6gl9 A 1.7 BS01 F3W A 1 L828 V836 A853 Y904 L905 C909 R911 R953 L956 L17 V25 A42 Y93 L94 C98 R100 R142 L145 A949 A951 R953 N954 D967 A138 A140 R142 N143 D156 2.7.10.2 0004672,0005524,0006468 ic50=135nM -logKd/Ki=6.87, Kd=135nM IC50=135nM P52333 29852068 1201 QDPTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRALAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR 6gl9 A 1.7 BS02 PHU A 1 W1011 M1037 R1059 L1060 W1078 W200 M226 R248 L249 W267 A949 A951 R953 N954 D967 A138 A140 R142 N143 D156 2.7.10.2 0004672,0005524,0006468 P52333 29852068 1202 QDPTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRALAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR 6gl9 B 1.7 BS01 F3W B 1 L828 V836 A853 Y904 L905 C909 R911 D912 R953 L956 L16 V24 A41 Y92 L93 C97 R99 D100 R141 L144 A949 A951 R953 N954 D967 A137 A139 R141 N142 D155 2.7.10.2 0004672,0005524,0006468 ic50=135nM IC50=135nM P52333 29852068 1201 DPTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRALAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR 6gl9 B 1.7 BS02 PHU B 1 W1011 M1037 R1059 L1060 W1078 W199 M225 R247 L248 W266 A949 A951 R953 N954 D967 A137 A139 R141 N142 D155 2.7.10.2 0004672,0005524,0006468 P52333 29852068 1202 DPTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRALAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR