6gbx A 1.72 BS01 ZN A 1 D159 E202 H330 D126 E169 H297 2.3.2.5 0005515,0005576,0008270,0016603,0016746,0017186,0035580,0036211,0046872,0070062,1904724,1904813 Q16769 30132075 401 SAWPEEKNYHQPAILNSSALRQIAEGTSISEMWQNDLQPLLIERYPGSPGSYAARQHIMQRIQRLQADWVLEIDTFLSQTPEGERSFSNIISTLNPTAKRHLVLACHYDSKYFSHWNNRVFVGATDSAVPCAMMLELARALDKKLLSLKTVSDSKPDLSLQLIFFDGEEAFLHWSPQDSLYGSRHLAAKMASTPHPPGARGTSQLHGMDLLVLLDLIGAPNPTFPNFFPNSARWFERLQAIEHELHELGLLKDHSLEGRYFQNYSYGGVIQDDHIPFLRRGVPVLHLIPSPFPEVWHTMDDNEENLDESTIDNLNKILQVFVLEYLHL 6gbx A 1.72 BS02 S77 A 1 K144 D159 E201 W207 D248 Q304 D305 W329 H330 K111 D126 E168 W174 D215 Q271 D272 W296 H297 2.3.2.5 0005515,0005576,0008270,0016603,0016746,0017186,0035580,0036211,0046872,0070062,1904724,1904813 Ki=0.02uM -logKd/Ki=7.70, Ki=0.020uM IC50=17nM Q16769 30132075 403 SAWPEEKNYHQPAILNSSALRQIAEGTSISEMWQNDLQPLLIERYPGSPGSYAARQHIMQRIQRLQADWVLEIDTFLSQTPEGERSFSNIISTLNPTAKRHLVLACHYDSKYFSHWNNRVFVGATDSAVPCAMMLELARALDKKLLSLKTVSDSKPDLSLQLIFFDGEEAFLHWSPQDSLYGSRHLAAKMASTPHPPGARGTSQLHGMDLLVLLDLIGAPNPTFPNFFPNSARWFERLQAIEHELHELGLLKDHSLEGRYFQNYSYGGVIQDDHIPFLRRGVPVLHLIPSPFPEVWHTMDDNEENLDESTIDNLNKILQVFVLEYLHL 6gbx B 1.72 BS01 ZN B 1 D159 E202 H330 D126 E169 H297 2.3.2.5 0005515,0005576,0008270,0016603,0016746,0017186,0035580,0036211,0046872,0070062,1904724,1904813 Q16769 30132075 401 SAWPEEKNYHQPAILNSSALRQIAEGTSISEMWQNDLQPLLIERYPGSPGSYAARQHIMQRIQRLQADWVLEIDTFLSQTPEGERSFSNIISTLNPTAKRHLVLACHYDSKYFSHWNNRVFVGATDSAVPCAMMLELARALDKKLLSLKTVSDSKPDLSLQLIFFDGEEAFLHWSPQDSLYGSRHLAAKMASTPHPPGARGTSQLHGMDLLVLLDLIGAPNPTFPNFFPNSARWFERLQAIEHELHELGLLKDHSLEGRYFQNYSYGGVIQDDHIPFLRRGVPVLHLIPSPFPEVWHTMDDNEENLDESTIDNLNKILQVFVLEYLHL 6gbx B 1.72 BS02 S77 B 1 K144 D159 E201 W207 D248 Q304 D305 W329 H330 K111 D126 E168 W174 D215 Q271 D272 W296 H297 2.3.2.5 0005515,0005576,0008270,0016603,0016746,0017186,0035580,0036211,0046872,0070062,1904724,1904813 Ki=0.02uM IC50=17nM Q16769 30132075 403 SAWPEEKNYHQPAILNSSALRQIAEGTSISEMWQNDLQPLLIERYPGSPGSYAARQHIMQRIQRLQADWVLEIDTFLSQTPEGERSFSNIISTLNPTAKRHLVLACHYDSKYFSHWNNRVFVGATDSAVPCAMMLELARALDKKLLSLKTVSDSKPDLSLQLIFFDGEEAFLHWSPQDSLYGSRHLAAKMASTPHPPGARGTSQLHGMDLLVLLDLIGAPNPTFPNFFPNSARWFERLQAIEHELHELGLLKDHSLEGRYFQNYSYGGVIQDDHIPFLRRGVPVLHLIPSPFPEVWHTMDDNEENLDESTIDNLNKILQVFVLEYLHL 6gbx C 1.72 BS01 ZN C 1 D159 E202 H330 D126 E169 H297 2.3.2.5 0005515,0005576,0008270,0016603,0016746,0017186,0035580,0036211,0046872,0070062,1904724,1904813 Q16769 30132075 401 SAWPEEKNYHQPAILNSSALRQIAEGTSISEMWQNDLQPLLIERYPGSPGSYAARQHIMQRIQRLQADWVLEIDTFLSQTPEGERSFSNIISTLNPTAKRHLVLACHYDSKYFSHWNNRVFVGATDSAVPCAMMLELARALDKKLLSLKTVSDSKPDLSLQLIFFDGEEAFLHWSPQDSLYGSRHLAAKMASTPHPPGARGTSQLHGMDLLVLLDLIGAPNPTFPNFFPNSARWFERLQAIEHELHELGLLKDHSLEGRYFQNYSYGGVIQDDHIPFLRRGVPVLHLIPSPFPEVWHTMDDNEENLDESTIDNLNKILQVFVLEYLHL 6gbx C 1.72 BS02 S77 C 1 K144 D159 E201 W207 D248 Q304 D305 W329 H330 K111 D126 E168 W174 D215 Q271 D272 W296 H297 2.3.2.5 0005515,0005576,0008270,0016603,0016746,0017186,0035580,0036211,0046872,0070062,1904724,1904813 Ki=0.02uM IC50=17nM Q16769 30132075 403 SAWPEEKNYHQPAILNSSALRQIAEGTSISEMWQNDLQPLLIERYPGSPGSYAARQHIMQRIQRLQADWVLEIDTFLSQTPEGERSFSNIISTLNPTAKRHLVLACHYDSKYFSHWNNRVFVGATDSAVPCAMMLELARALDKKLLSLKTVSDSKPDLSLQLIFFDGEEAFLHWSPQDSLYGSRHLAAKMASTPHPPGARGTSQLHGMDLLVLLDLIGAPNPTFPNFFPNSARWFERLQAIEHELHELGLLKDHSLEGRYFQNYSYGGVIQDDHIPFLRRGVPVLHLIPSPFPEVWHTMDDNEENLDESTIDNLNKILQVFVLEYLHL