6g31 A 3.0 BS01 ZOL A 1 D64 R73 D60 R69 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 QETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 A 3.0 BS02 MG A 1 D64 D68 D60 D64 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 QETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 A 3.0 BS03 MG A 2 D64 D68 D60 D64 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 QETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 B 3.0 BS01 ZOL B 1 D64 D68 R73 D59 D63 R68 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 B 3.0 BS02 MG B 1 D64 D68 D59 D63 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 B 3.0 BS03 MG B 2 D64 D68 D59 D63 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 C 3.0 BS01 ZOL C 1 D64 D68 R73 Q126 K151 D61 D65 R70 Q123 K148 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 TQETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSNKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 C 3.0 BS02 MG C 1 D64 D68 D61 D65 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 TQETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSNKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 C 3.0 BS03 MG C 2 D64 D68 D61 D65 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 TQETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSNKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 D 3.0 BS01 ZOL D 1 D64 D68 R73 D55 D59 R64 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 ETVQRILLEPYKYLLQLPGTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMF 6g31 D 3.0 BS02 MG D 1 D64 D68 D55 D59 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 ETVQRILLEPYKYLLQLPGTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMF 6g31 D 3.0 BS03 MG D 2 D64 D68 D55 D59 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 ETVQRILLEPYKYLLQLPGTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMF 6g31 E 3.0 BS01 ZOL E 1 D64 D68 R73 D49 D53 R58 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 QETVQRILLEPYKYLLQLAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPTQVQNILRQRTENIDIKKYCVHYGSFEYTRNTLKELEAKPELVALVKHLSKMFK 6g31 E 3.0 BS02 MG E 1 D64 D68 D49 D53 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 QETVQRILLEPYKYLLQLAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPTQVQNILRQRTENIDIKKYCVHYGSFEYTRNTLKELEAKPELVALVKHLSKMFK 6g31 E 3.0 BS03 MG E 2 D64 D68 D49 D53 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 QETVQRILLEPYKYLLQLAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPTQVQNILRQRTENIDIKKYCVHYGSFEYTRNTLKELEAKPELVALVKHLSKMFK 6g31 F 3.0 BS01 ZOL F 1 D64 D68 R73 Q126 D59 D63 R68 Q121 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 F 3.0 BS02 MG F 1 D64 D68 D59 D63 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 G 3.0 BS01 ZOL G 1 D64 Q126 K151 D62 Q124 K149 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 KTQETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKPLLNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMF 6g31 G 3.0 BS02 MG G 1 D64 D68 D62 D66 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 KTQETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKPLLNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMF 6g31 G 3.0 BS03 MG G 2 D64 D68 D62 D66 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 KTQETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKPLLNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMF 6g31 H 3.0 BS01 ZOL H 1 D64 D68 K212 D57 D61 K197 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 ETVQRILLEPYKYLLQLPQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 H 3.0 BS02 MG H 1 D64 D68 D57 D61 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 ETVQRILLEPYKYLLQLPQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 H 3.0 BS03 MG H 2 D64 D68 D57 D61 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 ETVQRILLEPYKYLLQLPQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 I 3.0 BS01 ZOL I 1 D64 K151 D60 K147 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 QETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLKSFCEDLTEGKFSFPTIHAIWSRPEVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDGNPELVALVKHLSKM 6g31 I 3.0 BS02 MG I 1 D64 D68 D60 D64 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 QETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLKSFCEDLTEGKFSFPTIHAIWSRPEVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDGNPELVALVKHLSKM 6g31 I 3.0 BS03 MG I 2 D64 D68 D60 D64 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 QETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLKSFCEDLTEGKFSFPTIHAIWSRPEVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDGNPELVALVKHLSKM 6g31 J 3.0 BS01 ZOL J 1 D64 D68 D59 D63 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 J 3.0 BS02 MG J 1 D64 D68 D59 D63 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 J 3.0 BS03 MG J 2 D64 D68 D59 D63 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 K 3.0 BS01 ZOL K 1 D64 D68 Q126 D60 D64 Q122 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 QETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKKPLLNTLGLFFQIRYDYANLHSSFCEDLTEGKFSFPTIHAIWSRPEQVQNILRQRTENIDIKKYCVHYLEDVGYTRNTLKELEAKAYKQPELVALVKHLSKMF 6g31 K 3.0 BS02 MG K 1 D64 D68 D60 D64 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 QETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKKPLLNTLGLFFQIRYDYANLHSSFCEDLTEGKFSFPTIHAIWSRPEQVQNILRQRTENIDIKKYCVHYLEDVGYTRNTLKELEAKAYKQPELVALVKHLSKMF 6g31 K 3.0 BS03 MG K 2 D64 D68 Q126 D60 D64 Q122 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 QETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKKPLLNTLGLFFQIRYDYANLHSSFCEDLTEGKFSFPTIHAIWSRPEQVQNILRQRTENIDIKKYCVHYLEDVGYTRNTLKELEAKAYKQPELVALVKHLSKMF 6g31 L 3.0 BS01 ZOL L 1 D64 D68 D59 D63 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 IC50=100000nM, Ki=2700nM O95749 30275041 401 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 L 3.0 BS02 MG L 1 D64 D68 D59 D63 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 403 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6g31 L 3.0 BS03 MG L 2 D64 D68 K212 D59 D63 K199 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 O95749 30275041 404 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRYDYANLHSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK