6fyp A 2.29 BS01 3NG A 1 L162 G163 E164 F167 V170 A184 K186 V220 F236 L239 N242 L290 D320 L28 G29 E30 F33 V36 A50 K52 V86 F102 L105 N108 L156 D186 2.7.12.1 0004672,0005524,0006468 ic50=143nM -logKd/Ki=6.84, IC50=143nM IC50=41nM P49761 29985556 501 SVEDDKEGHLVCRIGDWLQERYEIVGNLGEGTFGKVVECLDHARGKSQVALKIIRNVGKYREAARLEINVLKKIKEKDKENKFLCVLMSDWFNFHGHMCIAFELLGKNTFEFLKENNFQPYPLPHVRHMAYQLCHALRFLHENQLTHTDLKPENILFVNSEFETLYNEHKSCEEKSVKNTSIRVADFGSATFDHEHHTTIVATRHYRPPEVILELGWAQPCDVWSIGCILFEYYRGFTLFQTHENREHLVMMEKILGPIPSHMIHRTRKQKYFYKGGLVWDENSSDGRYVKENCKPLKSYMLQDSLEHVQLFDLMRRMLEFDPAQRITLAEALLHPFFAGLTPEERSF