6eum A 1.18 BS01 ZN A 1 D120 C198 H240 D85 C163 H205 H116 H118 D120 H179 C198 K201 N210 H240 H81 H83 D85 H144 C163 K166 N175 H205 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 P04190 29655609 301 KTVIKNETGTISISQLNKNVWVHTELGSFNGEAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 6eum A 1.18 BS02 ZN A 2 H116 H118 H179 H81 H83 H144 H116 H118 D120 H179 C198 K201 N210 H240 H81 H83 D85 H144 C163 K166 N175 H205 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 P04190 29655609 302 KTVIKNETGTISISQLNKNVWVHTELGSFNGEAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 6eum A 1.18 BS03 BY5 A 1 W89 H118 D120 H179 C198 N210 H240 W54 H83 D85 H144 C163 N175 H205 H116 H118 D120 H179 C198 K201 N210 H240 H81 H83 D85 H144 C163 K166 N175 H205 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=0.3uM -logKd/Ki=6.52, IC50=0.3uM IC50=300nM P04190 29655609 304 KTVIKNETGTISISQLNKNVWVHTELGSFNGEAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK