6es0 A 2.38 BS01 BW8 A 1 R26 A45 K47 E66 L70 L79 T95 Y97 M98 H144 L153 A163 D164 F165 W170 R22 A41 K43 E62 L66 L75 T91 Y93 M94 H140 L149 A159 D160 F161 W166 D146 Q150 N151 D164 D142 Q146 N147 D160 2.7.10.2,2.7.11.1 0004672,0005524,0006468 ic50=2.26uM -logKd/Ki=5.65, IC50=2.26uM IC50=4870nM O43353 29409752 401 AICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLHIHTPLLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLSKWGTIIYMPPENYASIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLKKTKLQS 6es0 B 2.38 BS01 BW8 B 1 R26 A45 K47 E66 L70 L79 T95 Y97 M98 H144 A163 D164 F165 K169 R22 A41 K43 E54 L58 L67 T83 Y85 M86 H132 A151 D152 F153 K157 D146 Q150 N151 D164 D134 Q138 N139 D152 2.7.10.2,2.7.11.1 0004672,0005524,0006468 ic50=2.26uM IC50=4870nM O43353 29409752 401 AICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLSKWRGTIIYMPPENYEPGQKSRASIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLKKTKLQ