6ehh A 2.4 BS01 2GE A 1 L9 F27 N33 F72 F74 M81 W117 D119 D120 F139 L8 F26 N32 F71 F73 M80 W116 D118 D119 F138 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=32nM -logKd/Ki=7.49, IC50=32nM P53368 29281266 201 STSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVDS 6ehh B 2.4 BS01 2GE B 1 F27 N33 F72 F74 W117 D119 D120 F139 F25 N31 F70 F72 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=32nM P53368 29281266 201 TSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVD 6ehh B 2.4 BS02 CU B 1 H90 H92 H88 H90 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 P53368 29281266 202 TSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVD 6ehh C 2.4 BS01 2GE C 1 N33 F72 F74 W117 D119 D120 F139 N31 F70 F72 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=32nM P53368 29281266 201 TSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVD 6ehh C 2.4 BS02 CU C 1 H90 H92 H88 H90 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 P53368 29281266 202 TSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVD 6ehh C 2.4 BS03 MG C 1 T63 D89 T61 D87 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 P53368 29281266 212 TSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVD 6ehh D 2.4 BS01 2GE D 1 L9 F27 N33 F72 F74 M81 W117 D119 D120 F139 L7 F25 N31 F70 F72 M79 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=32nM P53368 29281266 201 TSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVDSF 6ehh D 2.4 BS02 CU D 1 H90 H92 H88 H90 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 P53368 29281266 202 TSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVDSF