6dk1 A 3.12 BS01 GM4 A 1 V84 W89 Y103 F107 E172 F184 A185 V77 W82 Y96 F100 E165 F177 A178 ? 0004985,0005515,0005634,0005635,0005637,0005640,0005783,0005789,0005811,0005829,0005886,0006869,0007399,0014069,0016020,0030426,0031410,0038003,0038023,0042995,0043523,0045202,0045211,0070161,0070207,0098794,0098839,0098978,0150052 -logKd/Ki=7.65, Kd=22.5nM Ki=3.1nM, Kd=11.6nM, IC50=8.2nM Q99720 30291362 301 RWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSRLIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRYWAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPSTLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYLF 6dk1 B 3.12 BS01 GM4 B 1 V84 A86 W89 Y103 Y120 E172 A185 V85 A87 W90 Y104 Y121 E173 A186 ? 0004985,0005515,0005634,0005635,0005637,0005640,0005783,0005789,0005811,0005829,0005886,0006869,0007399,0014069,0016020,0030426,0031410,0038003,0038023,0042995,0043523,0045202,0045211,0070161,0070207,0098794,0098839,0098978,0150052 Ki=3.1nM, Kd=11.6nM, IC50=8.2nM Q99720 30291362 301 SMQWAVGRRWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSRLIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRYWAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPSTLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYLF 6dk1 C 3.12 BS01 GM4 C 1 V84 Y103 L105 F107 W164 E172 A185 V83 Y102 L104 F106 W163 E171 A184 ? 0004985,0005515,0005634,0005635,0005637,0005640,0005783,0005789,0005811,0005829,0005886,0006869,0007399,0014069,0016020,0030426,0031410,0038003,0038023,0042995,0043523,0045202,0045211,0070161,0070207,0098794,0098839,0098978,0150052 Ki=3.1nM, Kd=11.6nM, IC50=8.2nM Q99720 30291362 301 QWAVGRRWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSRLIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRYWAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPSTLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYLFGQ