6c91 B 2.895 BS01 EQD B 1 D149 M154 N162 F195 W223 T245 I247 D80 M85 N93 F116 W144 T166 I168 ? 0005524,0006457,0016887,0051082,0140662 Ki=440nM, IC50=1200nM P41148 29528635 405 REKSEKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSEDGQSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTTVWDWELMN 6c91 C 2.895 BS01 EQD C 1 N107 D149 M154 N162 F195 I247 N34 D76 M81 N89 F109 I161 ? 0005524,0006457,0016887,0051082,0140662 -logKd/Ki=6.19, Kd=0.65uM Ki=440nM, IC50=1200nM P41148 29528635 403 EKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSQSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTGGGGKTVWDWELMN