6bkw A 1.499 BS01 DXM A 1 L408 T410 G411 F413 V416 K430 Y476 M477 G480 N526 L528 D539 Y551 L16 T18 G19 F21 V24 K38 Y84 M85 G88 N134 L136 D147 Y159 D521 R525 N526 D539 D129 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=8.30, IC50=5nM Q06187 30756207 704 GSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN 6bkw A 1.499 BS02 FPZ A 1 W395 W421 Y425 Y461 W3 W29 Y33 Y69 D521 R525 N526 D539 D129 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 Q06187 30756207 705 GSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN