6ax1 A 2.26 BS01 C0S A 1 G50 A51 S122 M123 N152 G33 A34 S105 M106 N135 3.1.1.23 0004622,0005515,0005737,0005789,0005829,0005886,0006629,0006633,0006639,0006954,0009966,0016020,0016042,0019369,0019433,0042803,0046464,0047372,0050727,0051930,0052651,0052689,2000124 -logKd/Ki=9.42, IC50=0.38nM IC50=0.380000nM Q99685 29148769 401 DLPHLVNADGQYLFCRYWKPTGTPKALIFVSHGAGEHSGRYEELARMLMGLDLLVFAHDHVGHGQSEGERMVVSDFHVFVRDVLQHVDSMQKDYPGLPVFLLGHSMGGAIAILTAAERPGHFAGMVLISPLVLANPESATTFKVLAAKVLNLVLPNLSLGPIDSSVLSRNKTEVDIYNSDPLICRAGLKVCFGIQLLNAVSRVERALPKLTVPFLLLQGSADRLCDSKGAYLLMELAKSQDKTLKIYEGAYHVLHKELPEVTNSVFHEINMWVSQRTATA 6ax1 A 2.26 BS02 GOL A 1 G50 A51 H121 H269 G33 A34 H104 H252 3.1.1.23 0004622,0005515,0005737,0005789,0005829,0005886,0006629,0006633,0006639,0006954,0009966,0016020,0016042,0019369,0019433,0042803,0046464,0047372,0050727,0051930,0052651,0052689,2000124 Q99685 29148769 402 DLPHLVNADGQYLFCRYWKPTGTPKALIFVSHGAGEHSGRYEELARMLMGLDLLVFAHDHVGHGQSEGERMVVSDFHVFVRDVLQHVDSMQKDYPGLPVFLLGHSMGGAIAILTAAERPGHFAGMVLISPLVLANPESATTFKVLAAKVLNLVLPNLSLGPIDSSVLSRNKTEVDIYNSDPLICRAGLKVCFGIQLLNAVSRVERALPKLTVPFLLLQGSADRLCDSKGAYLLMELAKSQDKTLKIYEGAYHVLHKELPEVTNSVFHEINMWVSQRTATA 6ax1 A 2.26 BS03 GOL A 2 K165 I211 K148 I194 3.1.1.23 0004622,0005515,0005737,0005789,0005829,0005886,0006629,0006633,0006639,0006954,0009966,0016020,0016042,0019369,0019433,0042803,0046464,0047372,0050727,0051930,0052651,0052689,2000124 Q99685 29148769 403 DLPHLVNADGQYLFCRYWKPTGTPKALIFVSHGAGEHSGRYEELARMLMGLDLLVFAHDHVGHGQSEGERMVVSDFHVFVRDVLQHVDSMQKDYPGLPVFLLGHSMGGAIAILTAAERPGHFAGMVLISPLVLANPESATTFKVLAAKVLNLVLPNLSLGPIDSSVLSRNKTEVDIYNSDPLICRAGLKVCFGIQLLNAVSRVERALPKLTVPFLLLQGSADRLCDSKGAYLLMELAKSQDKTLKIYEGAYHVLHKELPEVTNSVFHEINMWVSQRTATA 6ax1 B 2.26 BS01 C0S B 1 A51 S122 M123 A46 S117 M118 3.1.1.23 0004622,0005515,0005737,0005789,0005829,0005886,0006629,0006633,0006639,0006954,0009966,0016020,0016042,0019369,0019433,0042803,0046464,0047372,0050727,0051930,0052651,0052689,2000124 IC50=0.380000nM Q99685 29148769 401 SPRRTPQSIPYQDLPHLVNADGQYLFCRYWKPTGTPKALIFVSHGAGEHSGRYEELARMLMGLDLLVFAHDHVGHGQSEGERMVVSDFHVFVRDVLQHVDSMQKDYPGLPVFLLGHSMGGAIAILTAAERPGHFAGMVLISPLVLAKVLAAKVLNLVLPNLSLGPIDSSVLSRNKTEVDIYNSDPLICRAGLKVCFGIQLLNAVSRVERALPKLTVPFLLLQGSADRLCDSKGAYLLMELAKSQDKTLKIYEGAYHVLHKELPEVTNSVFHEINMWVSQRTAT 6ax1 B 2.26 BS02 GOL B 1 H121 L184 H269 H116 L171 H256 3.1.1.23 0004622,0005515,0005737,0005789,0005829,0005886,0006629,0006633,0006639,0006954,0009966,0016020,0016042,0019369,0019433,0042803,0046464,0047372,0050727,0051930,0052651,0052689,2000124 Q99685 29148769 402 SPRRTPQSIPYQDLPHLVNADGQYLFCRYWKPTGTPKALIFVSHGAGEHSGRYEELARMLMGLDLLVFAHDHVGHGQSEGERMVVSDFHVFVRDVLQHVDSMQKDYPGLPVFLLGHSMGGAIAILTAAERPGHFAGMVLISPLVLAKVLAAKVLNLVLPNLSLGPIDSSVLSRNKTEVDIYNSDPLICRAGLKVCFGIQLLNAVSRVERALPKLTVPFLLLQGSADRLCDSKGAYLLMELAKSQDKTLKIYEGAYHVLHKELPEVTNSVFHEINMWVSQRTAT