5zun A 1.35 BS01 9JX A 1 G50 A51 E53 R57 H121 S122 M123 I179 S181 S185 E190 V191 Y194 L205 L241 V270 K273 G44 A45 E47 R51 H115 S116 M117 I173 S175 S179 E184 V185 Y188 L199 L235 V264 K267 3.1.1.23 0004622,0005515,0005737,0005789,0005829,0005886,0006629,0006633,0006639,0006954,0009966,0016020,0016042,0019369,0019433,0042803,0046464,0047372,0050727,0051930,0052651,0052689,2000124 ic50=0.64nM -logKd/Ki=9.19, IC50=0.64nM IC50=0.640000nM Q99685 30251836 401 PRRTPQSIPYQDLPHLVNADGQYLFCRYWAPTGTPKALIFVSHGAGEHSGRYEELARMLMGLDLLVFAHDHVGHGQSEGERMVVSDFHVFVRDVLQHVDSMQKDYPGLPVFLLGHSMGGAIAILTAAERPGHFAGMVLISPLVLANPESATTFKVLAAKVLNSVLPNLSSGPIDSSVLSRNKTEVDIYNSDPLICRAGLKVCFGIQLLNAVSRVERALPKLTVPFLLLQGSADRLCDSKGAYLLMELAKSQDKTLKIYEGAYHVLHKELPEVTNSVFHEINMWVSQRTA