5z1r A 1.62 BS01 EFL A 1 W81 V87 L94 N140 I146 W49 V55 L62 N108 I114 ? -logKd/Ki=5.70, IC50=1.99uM IC50=1990nM O60885 29541371 201 HHHHHLVPRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT