5yu9 A 1.95 BS01 1E8 A 1 L718 G719 A743 K745 M766 M790 M793 C797 R841 L844 T854 D855 F856 L19 G20 A44 K46 M63 M87 M90 C94 R138 L141 T151 D152 F153 D837 A839 R841 N842 D855 D134 A136 R138 N139 D152 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=6.74, Kd=0.18uM IC50=0.5nM, Kd=6.9nM P00533 27626175 1101 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVDADEYL 5yu9 B 1.95 BS01 1E8 B 1 L718 A743 K745 M790 M793 C797 R841 L844 T854 D855 L20 A45 K47 M87 M90 C94 R138 L141 T151 D152 D837 A839 R841 N842 D855 D134 A136 R138 N139 D152 2.7.10.1 0004672,0004713,0005524,0006468 IC50=0.5nM, Kd=6.9nM P00533 27626175 1101 PNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVV 5yu9 C 1.95 BS01 1E8 C 1 V726 A743 M790 M793 G796 C797 D800 T854 D855 F856 V30 A47 M90 M93 G96 C97 D100 T154 D155 F156 D837 A839 R841 N842 D855 D137 A139 R141 N142 D155 2.7.10.1 0004672,0004713,0005524,0006468 IC50=0.5nM, Kd=6.9nM P00533 27626175 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMVDADEYLIPQQ 5yu9 D 1.95 BS01 1E8 D 1 V726 A743 K745 M790 M793 G796 C797 D800 T854 D855 V27 A44 K46 M91 M94 G97 C98 D101 T155 D156 D837 A839 R841 N842 D855 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 IC50=0.5nM, Kd=6.9nM P00533 27626175 1101 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVD