5yfs A 2.3 BS01 RI2 A 1 M19 R22 G23 A24 R65 S137 K138 A139 D204 N214 K215 K240 F281 M17 R20 G21 A22 R63 S135 K136 A137 D202 N212 K213 K238 F279 5.3.1.29 0016853,0019323,0019509,0043917,0044237,0044249,0046523 Kd=13.8uM -logKd/Ki=4.86, Kd=13.8uM O57947 29382938 401 AMIVKEVYETAEKIKSMEIRGAGRIARAAAQALMIQAEKSKAKEPEELWNELKVASKILYNTRPTAVSLPNALRYVMHRVKAAYLGGADLETLRFTAINSAKEFIYNSEKAIERIGEIGAKRIEDGDIIMTHSHSKAAISVMKKAFEQGKNIKVIVTETRPKWQGKITAKELASYGIPVIYIVDSAARHYMKMTDKVVMGADSITANGAVINKIGTSLIALTAKEHRVWVMIAAETYKFHPATMLGQLVEIEMRDPTEVIPEEELRTWPKNIEVWNPAFDVTPPEYIDVIITERGIIPPYAAIDILKEEFGWALKYKEPWED 5yfs B 2.3 BS01 RI2 B 1 R22 G23 A24 G25 R65 S137 K138 A139 Q166 A203 D204 N214 K215 K240 F281 R20 G21 A22 G23 R63 S135 K136 A137 Q164 A201 D202 N212 K213 K238 F279 5.3.1.29 0016853,0019323,0019509,0043917,0044237,0044249,0046523 Kd=13.8uM O57947 29382938 401 AMIVKEVYETAEKIKSMEIRGAGRIARAAAQALMIQAEKSKAKEPEELWNELKVASKILYNTRPTAVSLPNALRYVMHRVKAAYLGGADLETLRFTAINSAKEFIYNSEKAIERIGEIGAKRIEDGDIIMTHSHSKAAISVMKKAFEQGKNIKVIVTETRPKWQGKITAKELASYGIPVIYIVDSAARHYMKMTDKVVMGADSITANGAVINKIGTSLIALTAKEHRVWVMIAAETYKFHPATMLGQLVEIEMRDPTEVIPEEELRTWPKNIEVWNPAFDVTPPEYIDVIITERGIIPPYAAIDILKEEFGWALKYKEPWED 5yfs C 2.3 BS01 RI2 C 1 R22 G23 A24 G25 R65 S137 K138 A139 D204 N214 K215 K240 F281 R20 G21 A22 G23 R63 S135 K136 A137 D202 N212 K213 K238 F279 5.3.1.29 0016853,0019323,0019509,0043917,0044237,0044249,0046523 Kd=13.8uM O57947 29382938 401 AMIVKEVYETAEKIKSMEIRGAGRIARAAAQALMIQAEKSKAKEPEELWNELKVASKILYNTRPTAVSLPNALRYVMHRVKAAYLGGADLETLRFTAINSAKEFIYNSEKAIERIGEIGAKRIEDGDIIMTHSHSKAAISVMKKAFEQGKNIKVIVTETRPKWQGKITAKELASYGIPVIYIVDSAARHYMKMTDKVVMGADSITANGAVINKIGTSLIALTAKEHRVWVMIAAETYKFHPATMLGQLVEIEMRDPTEVIPEEELRTWPKNIEVWNPAFDVTPPEYIDVIITERGIIPPYAAIDILKEEFGWALKYKEPWED