5y86 A 1.9 BS01 HRM A 1 A236 K238 F288 L291 L342 I354 A99 K101 F151 L154 L205 I217 D335 K337 N340 D355 S372 D198 K200 N203 D218 S235 2.7.12.1 0000242,0000287,0004672,0004674,0004712,0004713,0005524,0005634,0005654,0005737,0005813,0005829,0005856,0006468,0010494,0016310,0016607,0030218,0035063,0035617,0043066,0043231,0043518,0046872,0051301,0080135,0106310,1902751,1903008,1903432 ic50=0.8uM -logKd/Ki=6.10, IC50=0.8uM IC50=800nM O43781 29634919 601 VVPLTPEQALKQYKHHLTAYEKLEIINYPEIYFVGPNAKKRHGVIGGPNNGGYDDADGAYIHVPRDHLAYRYEVLKIIGKGSFGQVARVYDHKLRQYVALKMVRNEKRFHRQAAEEIRILEHLKKQDKTGSMNVIHMLESFTFRNHVCMAFELLSIDLYELIKKNKFQGFSVQLVRKFAQSILQSLDALHKNKIIHCDLKPENILLKHHGRSSTKVIDFGSSCFEYQKLYTYIQSRFYRAPEIILGSRYSTPIDIWSFGCILAELLTGQPLFPGEDEGDQLACMMELLGMPPPKLLEQSKRAKYFINSKGIPRYCSVTTQADGRVVLVGGRSRRGKKRGPPGSKDWGTALKGCDDYLFIEFLKRCLHWDPSARLTPAQALRHPWISKSVPRPLTT