5y2i B 1.917 BS01 8KX B 1 E19 N20 F22 R90 L95 W115 R116 P123 E17 N18 F20 R88 L93 W113 R114 P121 H11 R62 E89 H186 H9 R60 E87 H184 5.4.2.11,5.4.2.4 0003824,0004082,0004619,0005515,0005576,0005737,0005829,0006094,0006096,0016020,0016787,0016853,0016868,0019901,0034774,0046538,0061621,0070062,1904813 IC50=13100nM, Ki=3910nM P18669 301 AYKLVLIRHGESAWNLENRFSGWYDADLSPAGHEEAKRGGQALRDAGYEFDICFTSVQKRAIRTLWTVLDAIDQMWLPVVRTWRLNERHYGGLTGLNKAETAAKHGEAQVKIWRRSYDVPPPPMEPDHPFYSNISKDRRYADLTEDQLPSCESLKDTIARALPFWNEEIVPQIKEGKRVLIAAHGNSLRGIVKHLEGLSEEAIMELNLPTGIPIVYELDKNLKPIKPMQFLGD