5xdl A 2.7 BS01 8JC A 1 L718 V726 L792 M793 P794 G796 C797 R841 L844 L23 V31 L95 M96 P97 G99 C100 R144 L147 D837 R841 N842 D855 D140 R144 N145 D158 2.7.10.1 0004672,0004713,0005524,0006468 IC50=20nM, Ki=74nM, EC50=1655nM P00533 28881827 1101 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKEEATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPEDMDDVVDADEYLI