5wvd A 3.0 BS01 7UX A 1 E53 L55 L108 K126 L127 Q128 G129 L177 D191 F192 E13 L15 L68 K86 L87 Q88 G89 L137 D151 F152 D170 K172 N175 D191 D130 K132 N135 D151 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=7.68, IC50=21nM Q9BUB5 29497019 402 PGKFEDMYKLTSELLGEGAYAKVQGAVSLQNGKEYAVKIIEKQAGHSRSRVFREVETLYQCQGNKNILELIEFFEDDTRFYLVFEKLQGGSILAHIQKQKHFNEREASRVVRDVAAALDFLHTKGIAHRDLKPENILCESPEKVSPVKICDFDLGSGYMAPEVVEVFTDQATFYDKRCDLWSLGVVLYIMLSGYPPFKYEFPDKDWAHISSEAKDLISKLLVRDAKQRLSAAQVLQHPWVQ 5wvd B 3.0 BS01 7UX B 1 L55 V63 L108 L127 G129 L177 D191 F192 L15 V23 L68 L87 G89 L128 D140 F141 D170 K172 N175 D191 D121 K123 N126 D140 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=7.68, IC50=21nM Q9BUB5 29497019 401 PGKFEDMYKLTSELLGEGAYAKVQGAVSLQNGKEYAVKIIEKQAGHSRSRVFREVETLYQCQGNKNILELIEFFEDDTRFYLVFEKLQGGSILAHIQASRVVRDVAAALDFLHTKGIAHRDLKPENILCESPVSPVKICDFDLGSGMEYMAPEVVEVFTDQATFYDKRCDLWSLGVVLYIMLSGYPDLISKLLVRDAKQRLSAAQVLQHPWV