5wbz A 2.4 BS01 A4J A 1 N107 A224 A226 E227 P246 A256 G257 F260 G286 C289 N105 A222 A224 E225 P244 A254 G255 F258 G284 C287 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0016310,0032868,0042802,0042803,0046835,0070061,0070062,0070873 ic50=0.39uM -logKd/Ki=6.41, IC50=0.39uM IC50=450nM P50053 28853885 301 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbz B 2.4 BS01 A4J B 1 A224 A226 E227 T253 G257 C289 A227 A229 E230 T256 G260 C292 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0016310,0032868,0042802,0042803,0046835,0070061,0070062,0070873 ic50=0.39uM -logKd/Ki=6.41, IC50=0.39uM IC50=450nM P50053 28853885 301 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV