5w86 A 2.61 BS01 9YV A 1 L828 A853 M902 E903 L905 G908 L956 L15 A37 M80 E81 L83 G86 L134 D949 A951 R953 N954 D967 D127 A129 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=8.70, IC50=2nM IC50=2.0nM P52333 28947151 4000 PTIFEERHLKYISQLGKGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDML 5w86 B 2.61 BS01 9YV B 1 L828 V836 A853 V884 M902 E903 L905 G908 L956 L13 V18 A35 V66 M78 E79 L81 G84 L132 D949 A951 R953 N954 D967 D125 A127 R129 N130 D143 2.7.10.2 0004672,0004713,0005524,0006468 IC50=2.0nM P52333 28947151 4000 IFEERHLKYISQLGKGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDML 5w86 C 2.61 BS01 9YV C 1 Q827 L828 V836 A853 V884 M902 E903 L905 G908 L956 Q14 L15 V23 A40 V71 M84 E85 L87 G90 L138 D949 A951 R953 N954 D967 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 IC50=2.0nM P52333 28947151 4000 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLW 5w86 D 2.61 BS01 9YV D 1 L828 V836 A853 M902 E903 L905 G908 L956 L15 V23 A40 M82 E83 L85 G88 L136 D949 A951 R953 N954 D967 D129 A131 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 IC50=2.0nM P52333 28947151 4000 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQGPDQQRDFQREIQILKALHSDFIVKYRGVSYSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLW