5vry A 1.9 BS01 dna T 0 H34 S229 K230 G231 T233 K234 K280 R283 L287 T292 I293 N294 E295 Y296 H26 S221 K222 G223 T225 K226 K272 R275 L279 T284 I285 N286 E287 Y288 D190 D192 D256 D182 D184 D248 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 P06746 28682600 1 ~ 16 ETLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 5vry A 1.9 BS02 dna P 0 S104 G105 G107 P108 S109 A110 D190 D192 R254 D256 Y271 F272 T273 G274 D276 N279 S96 G97 G99 P100 S101 A102 D182 D184 R246 D248 Y263 F264 T265 G266 D268 N271 D190 D192 D256 D182 D184 D248 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 P06746 28682600 1 ~ 11 ETLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 5vry A 1.9 BS03 dna D 0 K35 A38 Y39 P63 G64 V65 G66 K68 I69 K27 A30 Y31 P55 G56 V57 G58 K60 I61 D190 D192 D256 D182 D184 D248 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 P06746 28682600 1 ~ 5 ETLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 5vry A 1.9 BS04 TTP P 1 G179 S180 R183 G189 D190 D192 Y271 F272 T273 G274 D276 N279 G171 S172 R175 G181 D182 D184 Y263 F264 T265 G266 D268 N271 D190 D192 D256 D182 D184 D248 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 IC50=1400nM P06746 28682600 101 ETLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 5vry A 1.9 BS05 MG P 1 D190 D192 D256 D182 D184 D248 D190 D192 D256 D182 D184 D248 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 P06746 28682600 103 ETLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 5vry A 1.9 BS06 MG P 2 D190 D192 D182 D184 D190 D192 D256 D182 D184 D248 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 P06746 28682600 104 ETLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 5vry A 1.9 BS07 MG P 3 T101 V103 I106 T93 V95 I98 D190 D192 D256 D182 D184 D248 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 P06746 28682600 105 ETLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE