5vcx A 2.7 BS01 H8H A 1 L116 A137 K139 T187 C190 F240 D251 L42 A63 K65 T113 C116 F166 D177 D233 K235 N238 D251 D270 D159 K161 N164 D177 D196 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=5.55, Kd=2817nM IC50=418nM, Ki=40nM, Kd=2817nM Q99640 28792760 401 HQLQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQ