5v24 A 2.5 BS01 8V7 A 1 L686 G687 K688 V694 K709 M754 Q756 V757 L810 D822 L16 G17 K18 V24 K39 M80 Q82 V83 L136 D148 D803 K805 D807 N808 D822 T842 D129 K131 D133 N134 D148 T159 2.7.11.25 0004672,0005524,0006468 ic50=400nM -logKd/Ki=6.40, IC50=400nM IC50=400nM Q99683 28291695 1000 LEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERDSPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLFTGTLQYMAPEIIDYGKAADIWSLGCTIIEMATGKPPFYEEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 5v24 B 2.5 BS01 8V7 B 1 G687 K688 V694 K709 M754 V757 L810 D822 G18 K19 V25 K40 M85 V88 L141 D153 D803 K805 D807 N808 D822 T842 D134 K136 D138 N139 D153 T165 2.7.11.25 0004672,0005524,0006468 ic50=400nM IC50=400nM Q99683 28291695 1000 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERDSRYSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLTFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLKV