5ura A 1.85002 BS01 8KS A 1 F17 M21 V26 T37 P39 S56 A76 D77 F105 M116 L118 Y129 F19 M23 V28 T39 P41 S58 A78 D79 F107 M118 L120 Y131 ? 0005504,0005515,0005634,0005737,0005829,0007399,0008285,0008289,0015908,0050673 Ki=0.4uM -logKd/Ki=6.40, Ki=0.4uM Ki=450nM O15540 28632393 201 SHMVEAFCATWKLTNSQNFDEYMKALGVGFATRQVGNVTKPTVIISQEGDKVVIRTLSTFKNTEISFQLGEEFDETTADDRNCKSVVSLDGDKLVHIQKWDGKETNFVREIKDGKMVMTLTFGDVVAVRHYEKA 5ura B 1.85002 BS01 8KS B 1 F17 M21 G34 P39 T54 S56 A76 D77 F105 M116 L118 Y129 F20 M24 G37 P42 T57 S59 A79 D80 F108 M119 L121 Y132 ? 0005504,0005515,0005634,0005737,0005829,0007399,0008285,0008289,0015908,0050673 Ki=0.4uM Ki=450nM O15540 28632393 201 GSHMVEAFCATWKLTNSQNFDEYMKALGVGFATRQVGNVTKPTVIISQEGDKVVIRTLSTFKNTEISFQLGEEFDETTADDRNCKSVVSLDGDKLVHIQKWDGKETNFVREIKDGKMVMTLTFGDVVAVRHYEKA 5ura C 1.85002 BS01 8KS C 1 F17 M21 G34 P39 S56 D77 F105 M116 L118 R127 Y129 F19 M23 G36 P41 S58 D79 F107 M118 L120 R129 Y131 ? 0005504,0005515,0005634,0005737,0005829,0007399,0008285,0008289,0015908,0050673 Ki=0.4uM Ki=450nM O15540 28632393 201 SHMVEAFCATWKLTNSQNFDEYMKALGVGFATRQVGNVTKPTVIISQEGDKVVIRTLSTFKNTEISFQLGEEFDETTADDRNCKSVVSLDGDKLVHIQKWDGKETNFVREIKDGKMVMTLTFGDVVAVRHYEKA 5ura D 1.85002 BS01 8KS D 1 F17 M21 T30 G34 T37 P39 S56 F58 D77 F105 M116 L118 R127 Y129 F19 M23 T32 G36 T39 P41 S58 F60 D79 F107 M118 L120 R129 Y131 ? 0005504,0005515,0005634,0005737,0005829,0007399,0008285,0008289,0015908,0050673 Ki=0.4uM Ki=450nM O15540 28632393 201 SHMVEAFCATWKLTNSQNFDEYMKALGVGFATRQVGNVTKPTVIISQEGDKVVIRTLSTFKNTEISFQLGEEFDETTADDRNCKSVVSLDGDKLVHIQKWDGKETNFVREIKDGKMVMTLTFGDVVAVRHYEKA