5ur1 A 2.2 BS01 YY9 A 1 L484 V492 K514 E531 M535 V561 A564 G567 L630 A640 D641 L21 V28 K50 E67 M71 V97 A100 G103 L161 A171 D172 D623 A625 R627 N628 D641 D154 A156 R158 N159 D172 2.7.10.1 0004672,0004713,0005007,0005524,0006468 ic50=1.06nM -logKd/Ki=8.97, IC50=1.06nM IC50=1.1nM P11362 28521156 801 ELPEDPRWELPRDRLVLGKPLGEGFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPYNPSHNPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 5ur1 B 2.2 BS01 YY9 B 1 V492 A512 K514 E531 I545 V561 Y563 A564 G567 L630 A640 D641 V29 A47 K49 E66 I80 V96 Y98 A99 G102 L150 A160 D161 D623 A625 R627 N628 D641 D143 A145 R147 N148 D161 2.7.10.1 0004672,0004713,0005007,0005524,0006468 ic50=1.06nM IC50=1.1nM P11362 28521156 801 ELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSN