5uiq A 2.64 BS01 8BV A 1 M192 V200 A211 Y262 M265 L318 M23 V31 A40 Y78 M81 L134 D311 K313 A315 N316 D329 T351 D127 K129 A131 N132 D145 T163 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 -logKd/Ki=4.26, IC50=55.056uM IC50=55000nM Q9NWZ3 28498658 501 RFHSFSFYELKNVTNNFDERPKMGEGGFGVVYKGYVTTVAVKKLAAKQQFDQEIKVMAKCQHENLVELLGFSSDCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 5uiq B 2.64 BS01 8BV B 1 V200 A211 Y262 Y264 M265 L318 V34 A43 Y86 Y88 M89 L142 D311 K313 A315 N316 D329 T351 D135 K137 A139 N140 D153 T170 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 IC50=55000nM Q9NWZ3 28498658 501 RFHSFSFYELKNVTNNFDERPIGNKMGEGGFGVVYKGYVTTVAVKKLAAEELKQQFDQEIKVMAKCQHENLVELLGFSSDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 5uiq C 2.64 BS01 8BV C 1 V200 A211 Y262 Y264 M265 L318 V37 A48 Y93 Y95 M96 L149 D311 K313 A315 N316 D329 T351 D142 K144 A146 N147 D160 T178 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 IC50=55000nM Q9NWZ3 28498658 501 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 5uiq D 2.64 BS01 8BV D 1 M192 V200 A211 Y262 M265 L318 M29 V35 A46 Y86 M89 L142 D311 K313 A315 N316 D329 T351 D135 K137 A139 N140 D153 T169 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 IC50=55000nM Q9NWZ3 28498658 501 RFHSFSFYELKNVTNNFDERPISVGGNKMGGFGVVYKGYVNNTTVAVKKLALKQQFDQEIKVMAKCQHENLVELLGFSSDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARATVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT