5sy3 A 2.3 BS01 74Z A 1 T18 Y20 V36 Y83 F119 F124 V127 T227 G228 A229 S230 T15 Y17 V33 Y80 F116 F121 V124 T220 G221 A222 S223 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D219 A222 3.4.23.15 0004190,0006508 ic50=43uM -logKd/Ki=4.37, IC50=43uM IC50=43000nM P00797 27687967 402 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR