5q14 A 1.85 BS01 peptide B 0 K307 I321 L324 K325 P467 L468 E471 K61 I75 L78 K79 P221 L222 E225 ? 0003677,0004879,0006355,0032052,0038183 Q96RI1 29204945 745 ~ 756 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q14 A 1.85 BS02 9MM A 1 I277 N287 M294 H298 M332 F333 R335 S336 I339 F340 I356 S359 M369 Y373 I31 N41 M48 H52 M86 F87 R89 S90 I93 F94 I110 S113 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 -logKd/Ki=7.68, IC50=0.021uM IC50=21nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q14 C 1.85 BS01 peptide D 0 V303 E304 K307 H317 I321 K325 P467 L468 E471 I472 V57 E58 K61 H71 I75 K79 P221 L222 E225 I226 ? 0003677,0004879,0006355,0032052,0038183 Q96RI1 29204945 746 ~ 756 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q14 C 1.85 BS02 9MM C 1 I273 I277 L291 M294 M332 F333 R335 S336 F340 I356 S359 Y373 M454 I27 I31 L45 M48 M86 F87 R89 S90 F94 I110 S113 Y127 M208 ? 0003677,0004879,0006355,0032052,0038183 IC50=21nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ