5oug A 2.57 BS01 L0B A 1 W53 L104 L106 Q114 L116 W54 L105 L107 Q115 L117 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 1101 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug A 2.57 BS02 9Z0 A 1 L54 I88 R96 L55 I89 R97 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 -logKd/Ki=2.77, Kd=1703.44uM 29237730 1104 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug A 2.57 BS03 9Z0 A 2 Y7 E9 L10 L63 Q64 Y70 V107 Y8 E10 L11 L64 Q65 Y71 V108 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 -logKd/Ki=2.77, Kd=1703.44uM 29237730 1105 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug A 2.57 BS04 L0B A 2 Y91 W145 T146 C186 Y92 W146 T147 C187 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 1106 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug A 2.57 BS05 9Z0 E 1 L100 T101 L101 T102 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 -logKd/Ki=2.77, Kd=1703.44uM 29237730 301 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug B 2.57 BS01 9Z0 A 1 L100 T101 L101 T102 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 1104 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug B 2.57 BS02 L0B A 2 W53 L106 Q114 L116 W54 L107 Q115 L117 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 1106 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug B 2.57 BS03 9Z0 B 1 I88 R96 P97 I89 R97 P98 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 306 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug B 2.57 BS04 9Z0 B 2 Y7 E9 L10 L63 Q64 V107 Y8 E10 L11 L64 Q65 V108 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 307 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug B 2.57 BS05 L0B B 1 Y91 W145 T146 Y184 Y92 W146 T147 Y185 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 308 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug C 2.57 BS01 L0B B 1 W53 L106 Q114 L116 W54 L107 Q115 L117 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 308 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug C 2.57 BS02 9Z0 C 1 L6 Y7 E9 L10 L63 V107 L7 Y8 E10 L11 L64 V108 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 305 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug C 2.57 BS03 L0B C 1 W145 T146 W146 T147 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 306 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug D 2.57 BS01 L0B C 1 W53 L104 L106 Q114 L116 W54 L105 L107 Q115 L117 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 306 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug D 2.57 BS02 9Z0 D 1 L90 R96 P97 Q121 L91 R97 P98 Q122 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 304 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug D 2.57 BS03 9Z0 D 2 Y7 E9 L10 Y62 L63 Q64 V107 Y8 E10 L11 Y63 L64 Q65 V108 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 305 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug D 2.57 BS04 L0B D 1 Y91 W145 T146 Y184 C186 Y92 W146 T147 Y185 C187 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 306 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug E 2.57 BS01 L0B A 1 Y91 W145 T146 Y184 Y92 W146 T147 Y185 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 1101 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug E 2.57 BS02 9Z0 D 1 L100 T101 P102 L101 T102 P103 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 304 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug E 2.57 BS03 L0B D 1 L36 W53 L104 L106 Q114 L116 L37 W54 L105 L107 Q115 L117 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 306 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug E 2.57 BS04 9Z0 E 1 I88 R96 P97 I89 R97 P98 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 301 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug E 2.57 BS05 9Z0 E 2 Y7 E9 L10 L63 Q64 Y70 V107 Y8 E10 L11 L64 Q65 Y71 V108 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 29237730 302 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG