5one A 2.6 BS01 9YQ A 1 L194 L210 E211 A213 G216 R220 L263 A273 L68 L84 E85 A87 G90 R94 L137 A147 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T158 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 -logKd/Ki=7.28, IC50=52nM EC50=38nM, IC50=52nM O14965 28818446 501 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS