5n4s A 1.2 BS01 ZN A 1 D118 C198 H240 D87 C167 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0046872 Q9K2N0 28470248 501 AYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5n4s A 1.2 BS02 ZN A 2 H114 H116 H179 H83 H85 H148 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0046872 Q9K2N0 28470248 502 AYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5n4s A 1.2 BS03 R38 A 1 Y67 H116 D118 H179 R205 G209 N210 H240 Y36 H85 D87 H148 R174 G178 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0046872 ic50=0.055uM -logKd/Ki=7.26, IC50=0.055uM Q9K2N0 28470248 504 AYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5n4s A 1.2 BS04 R38 B 1 G64 A65 G33 A34 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0046872 ic50=0.055uM -logKd/Ki=7.26, IC50=0.055uM Q9K2N0 28470248 504 AYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5n4s B 1.2 BS01 ZN B 1 D118 C198 H240 D86 C166 H208 H114 H116 D118 H179 C198 Y201 N210 H240 H82 H84 D86 H147 C166 Y169 N178 H208 3.5.2.6 0016787,0017001,0046872 Q9K2N0 28470248 501 AYPTVEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5n4s B 1.2 BS02 ZN B 2 H114 H116 H179 H82 H84 H147 H114 H116 D118 H179 C198 Y201 N210 H240 H82 H84 D86 H147 C166 Y169 N178 H208 3.5.2.6 0016787,0017001,0046872 Q9K2N0 28470248 502 AYPTVEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5n4s B 1.2 BS03 R38 B 1 Y67 H116 D118 H179 R205 N210 H240 Y35 H84 D86 H147 R173 N178 H208 H114 H116 D118 H179 C198 Y201 N210 H240 H82 H84 D86 H147 C166 Y169 N178 H208 3.5.2.6 0016787,0017001,0046872 ic50=0.055uM Q9K2N0 28470248 504 AYPTVEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR