5lhu A 2.02 BS01 HIS A 1 Y217 D218 L275 Y217 D218 L275 2.4.2.17 0000105,0000287,0003879,0005515,0005524,0005737,0005886,0016208,0016757,0046872 -logKd/Ki=4.66, IC50=22uM P9WMN1 28781362 301 MLRVAVPNKGALSEPATEILAEAGYRRRTDSKDLTVIDPVNNVEFFFLRPKDIAIYVGSGELDFGITGRDLVCDSGAQVRERLALGFGSSSFRYAAPAGRNWTTADLAGMRIATAYPNLVRKDLATKGIEATVIRLDGAVEISVQLGVADAIADVVGSGRTLSQHDLVAFGEPLCDSEAVLIERAGTDGQDQTEARDQLVARVQGVVFGQQYLMLDYDCPRSALKKATAITPGLESPTIAPLADPDWVAIRALVPRRDVNGIMDELAAIGAKAILASDIRFCRF