5lg3 A 3.567 BS01 Z80 A 1 I20 I23 F126 V147 T149 E155 D158 W160 I162 I10 I13 F116 V137 T139 E145 D148 W150 I152 ? 0004888,0005216,0005230,0006811,0007165,0016020,0034220,0042391,0042802,0043005 -logKd/Ki=3.80, IC50=158uM E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lg3 B 3.567 BS01 Z80 B 1 N21 I23 F126 V147 T149 E155 D158 W160 I162 N11 I13 F116 V137 T139 E145 D148 W150 I152 ? 0004888,0005216,0005230,0006811,0007165,0016020,0034220,0042391,0042802,0043005 -logKd/Ki=3.80, IC50=158uM E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lg3 C 3.567 BS01 Z80 C 1 N21 I23 F126 T149 E155 D158 W160 N11 I13 F116 T139 E145 D148 W150 ? 0004888,0005216,0005230,0006811,0007165,0016020,0034220,0042391,0042802,0043005 E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lg3 D 3.567 BS01 Z80 D 1 N21 I23 F126 T149 E155 D158 W160 I162 N11 I13 F116 T139 E145 D148 W150 I152 ? 0004888,0005216,0005230,0006811,0007165,0016020,0034220,0042391,0042802,0043005 E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lg3 E 3.567 BS01 Z80 E 1 I20 N21 I23 F126 T149 E150 E155 D158 W160 I10 N11 I13 F116 T139 E140 E145 D148 W150 ? 0004888,0005216,0005230,0006811,0007165,0016020,0034220,0042391,0042802,0043005 E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lg3 F 3.567 BS01 Z80 F 1 I20 I23 F126 V147 T149 E155 D158 W160 I162 I10 I13 F116 V137 T139 E145 D148 W150 I152 ? 0004888,0005216,0005230,0006811,0007165,0016020,0034220,0042391,0042802,0043005 E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lg3 G 3.567 BS01 Z80 G 1 I20 N21 I23 F126 V147 T149 N151 E155 D158 W160 I10 N11 I13 F116 V137 T139 N141 E145 D148 W150 ? 0004888,0005216,0005230,0006811,0007165,0016020,0034220,0042391,0042802,0043005 E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lg3 H 3.567 BS01 Z80 H 1 I20 I23 F126 V147 T149 E155 D158 W160 I162 I10 I13 F116 V137 T139 E145 D148 W150 I152 ? 0004888,0005216,0005230,0006811,0007165,0016020,0034220,0042391,0042802,0043005 E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lg3 I 3.567 BS01 Z80 I 1 N21 I23 F126 T149 E150 N151 E155 D158 W160 N11 I13 F116 T139 E140 N141 E145 D148 W150 ? 0004888,0005216,0005230,0006811,0007165,0016020,0034220,0042391,0042802,0043005 E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lg3 J 3.567 BS01 Z80 J 1 I20 I23 F126 V147 T149 E150 E155 W160 I10 I13 F116 V137 T139 E140 E145 W150 ? 0004888,0005216,0005230,0006811,0007165,0016020,0034220,0042391,0042802,0043005 E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI