5kx8 A 2.671 BS01 6YE A 1 M192 V200 A211 Y262 M265 G268 A315 N316 L318 S328 D329 M30 V38 A49 Y95 M98 G101 A148 N149 L151 S161 D162 D311 K313 A315 N316 D329 T351 D144 K146 A148 N149 D162 T180 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 -logKd/Ki=7.42, IC50=38nM IC50=38nM Q9NWZ3 27476420 501 TRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASETVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 5kx8 B 2.671 BS01 6YE B 1 M192 E194 V200 A211 Y262 Y264 M265 G268 N316 L318 S328 D329 M32 E34 V40 A51 Y90 Y92 M93 G96 N144 L146 S156 D157 D311 K313 A315 N316 D329 T351 D139 K141 A143 N144 D157 T173 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 IC50=38nM Q9NWZ3 27476420 501 SDTRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 5kx8 C 2.671 BS01 6YE C 1 M192 V200 A211 Y262 M265 G268 A315 L318 S328 D329 M29 V37 A48 Y96 M99 G102 A149 L152 S162 D163 D311 K313 A315 N316 D329 T351 D145 K147 A149 N150 D163 T181 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 IC50=38nM Q9NWZ3 27476420 501 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAAITTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASETVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTAS 5kx8 D 2.671 BS01 6YE D 1 M192 E194 G195 V200 A211 Y262 Y264 M265 G268 A315 N316 L318 S328 D329 M29 E31 G32 V37 A48 Y94 Y96 M97 G100 A147 N148 L150 S160 D161 D311 K313 A315 N316 D329 T351 D143 K145 A147 N148 D161 T178 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 IC50=38nM Q9NWZ3 27476420 501 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA