5ke0 A 1.68 BS01 6S9 A 1 G35 A50 K52 Q103 D104 L105 M106 E107 L154 D165 G20 A35 K37 Q88 D89 L90 M91 E92 L139 D150 D147 K149 S151 N152 D165 T188 D132 K134 S136 N137 D150 T173 2.7.11.24 0000165,0001784,0003690,0004672,0004674,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005769,0005770,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006974,0007166,0007507,0008284,0008286,0008353,0009636,0009887,0010759,0014032,0014044,0014069,0015966,0016020,0016301,0016310,0018105,0018107,0019233,0019858,0019901,0019902,0030278,0030335,0030424,0030521,0030641,0030878,0031143,0031435,0031647,0031663,0032212,0032355,0032496,0032839,0032872,0032991,0033574,0033598,0034198,0034614,0035094,0035556,0036120,0038127,0038133,0042220,0042307,0042473,0042542,0042552,0042802,0043204,0043330,0043401,0043627,0044849,0045596,0045727,0045893,0046697,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060045,0060291,0060324,0060425,0060440,0060716,0061308,0061431,0070161,0070371,0070849,0071276,0071320,0071356,0071364,0071380,0072584,0072686,0090170,0097237,0097305,0106310,0120041,1904355,1990314,2000641 -logKd/Ki=9.70, IC50=0.2nM IC50=0.200000nM P63086 27329786 401 VFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG