5ier A 2.005 BS01 3QZ A 1 L12 T43 A91 S93 F107 Y109 L11 T42 A90 S92 F106 Y108 -logKd/Ki=4.89, Kd~13uM 28980354 201 QSPALIASQSLWRCTQAHDREGWLALMADDVVIETPIGKSVTNPDGSGIKGKEAVGAFFDTHIAATRLTVTCEETFPSSSPDEIAHILVAHSEFDGGFTSEVRGVFTYRVNKAGLITNLRGYWNLDMMTFG 5ier B 2.005 BS01 3QZ B 1 L12 W13 T16 L69 A91 F107 L11 W12 T15 L68 A90 F106 28980354 201 QSPALIASQSLWRCTQAHDREGWLALMADDVVIETPIGKSVTNPDGSGIKGKEAVGAFFDTHIAATRLTVTCEETFPSSSPDEIAHILVAHSEFDGGFTSEVRGVFTYRVNKAGLITNLRGYWNLDMMTFG 5ier C 2.005 BS01 3QZ C 1 L12 T43 Y109 L11 T42 Y108 28980354 201 QSPALIASQSLWRCTQAHDREGWLALMADDVVIETPIGKSVTNPDGSGIKGKEAVGAFFDTHIAATRLTVTCEETFPSSSPDEIAHILVAHSEFDGGFTSEVRGVFTYRVNKAGLITNLRGYWNLDMMTFG 5ier D 2.005 BS01 3QZ D 1 L12 W13 V103 F107 L11 W12 V98 F102 28980354 201 QSPALIASQSLWRCTQAHDREGWLALMADDVVIETPIGKSVTNPDGSGIKGKEAVGAFFDTHIAATRLTVTCEETFPSSSPDEIAHILVAHSEFTSEVRGVFTYRVNKAGLITNLRGYWNLDMMTF