5i8b A 1.5218 BS01 ZN A 1 C1199 C1200 H1291 C1294 C121 C122 H205 C208 2.3.1.-,2.3.1.48 0004402,0006355 Q92793 27190605 1401 GSRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLGYCCGRKYEFSPQTLCCYGKQLCTIPRDAAYYSYQNRYHFCEKCFTLGDDPSQPQTTISKDQFEKKKNDTLDPEPFVDCKECGRKMHQICVLHYDIIWPSGFVCDNCL 5i8b A 1.5218 BS02 ZN A 2 C1283 C1286 C1308 C1311 C197 C200 C222 C225 2.3.1.-,2.3.1.48 0004402,0006355 Q92793 27190605 1402 GSRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLGYCCGRKYEFSPQTLCCYGKQLCTIPRDAAYYSYQNRYHFCEKCFTLGDDPSQPQTTISKDQFEKKKNDTLDPEPFVDCKECGRKMHQICVLHYDIIWPSGFVCDNCL 5i8b A 1.5218 BS03 ZN A 3 C1213 C1219 C135 C141 2.3.1.-,2.3.1.48 0004402,0006355 Q92793 27190605 1403 GSRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLGYCCGRKYEFSPQTLCCYGKQLCTIPRDAAYYSYQNRYHFCEKCFTLGDDPSQPQTTISKDQFEKKKNDTLDPEPFVDCKECGRKMHQICVLHYDIIWPSGFVCDNCL 5i8b A 1.5218 BS04 69F A 1 P1110 V1115 L1120 N1168 R1173 V1174 P32 V37 L42 N90 R95 V96 2.3.1.-,2.3.1.48 0004402,0006355 ic50=0.11uM -logKd/Ki=6.96, IC50=0.11uM EC50=>10000nM, IC50=110nM Q92793 27190605 1404 GSRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLGYCCGRKYEFSPQTLCCYGKQLCTIPRDAAYYSYQNRYHFCEKCFTLGDDPSQPQTTISKDQFEKKKNDTLDPEPFVDCKECGRKMHQICVLHYDIIWPSGFVCDNCL