5hi2 A 2.512 BS01 BAX A 1 A481 E501 L505 L514 T529 Q530 W531 C532 F583 G593 D594 F595 A33 E48 L52 L61 T76 Q77 W78 C79 F130 G140 D141 F142 D576 K578 N580 N581 D594 S616 D123 K125 N127 N128 D141 S145 2.7.11.1 0004672,0005524,0006468 IC50=22nM, Kd=260nM, Ki=22nM P15056 26996308 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLSILWMAPEVIRMNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELAREL